Exemever in the period of the steroid cycle prevents side effects that can cause flavoring steroids. It is worth noting that the action of Exemever is radically different from the action of the usual for many athletes Tamoxifen.
As is known, Tamoxifen does not exert any influence on the process of aromatization. It simply begins to interact with cellular estrogen receptors, not allowing estrogen to join them and form a bond.
Exemever acts on the process of aromatization and suppresses it. The structure of Exemever is very similar to the steroid of natural origin androstenedione. The principle of action of Exemever is that it irreversibly binds the active enzymes to hormones. As a result, hormones lose their activity. Exemever does not have non-estrogenic, non-progestogenic activity. But it is characterized by mild androgenic activity.
How to take Exemever
Exemever is a new generation drug that blocks enzymes responsible for aromatization. Exemever is called the real killer of aromatase. The principle of action of this drug is that it blocks the enzymes responsible for the synthesis of estrogens.
The amount of necessary exemestane is calculated taking into account the used anabolic steroids, individual sensitivity to aromatase inhibitors. In the most general case, the dosage of exemestane is 12.5 mg per day. It should be remembered that the use of exemestane serves only to control the desired level of estrogen. Complete reduction or removal of estrogens adversely affects the body.
The duration of taking the drug is 2-4 weeks. In the event that the athlete does not start taking aromatase inhibitors on time and already noticeable or even pronounced estrogenic side effects, you should begin taking 25 mg of Exemever daily and do not stop taking the drug until the signs of gynecomastia disappear completely.
It is recommended to take Exemever during meals or immediately after it. In this case, the bioavailability of the drug will increase by 40%, and within two hours its maximum concentration in the blood will be reached.
Take the drug can and athletes who suffer from liver or kidney disease. However, in this case, the systemic effect of the drug is increased by 2-3 times. Such athletes are recommended to reduce the dosage of Exemever.